SCHEMBL6753541

SCHEMBL6753541

NC1=CCCc2c(N)cccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
ALDH1A1 P00352 5/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CD44 P16070 1/20 0.36
HSD17B10 Q99714 2/20 0.32
CYP3A4 P08684 3/20 0.32
HPGD P15428 3/20 0.32
TSHR P16473 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
GID4 Q8IVV7 1/20 0.32
KDM4E B2RXH2 2/20 0.31
GAA P10253 2/20 0.31
PTPRC P08575 1/20 0.31
ADORA2A P29274 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
BRD4 O60885 1/20 0.31
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2212205 0.74 S100A4 (0.43) ALDH1A1L3MBTL1TSHRTDP1GAA
SCHEMBL19415422 0.71 PARP1 (0.42) PARP1ALDH1A1CD44
SCHEMBL29444072 0.70 NOS3 (0.45) PARP1ALDH1A1L3MBTL1HPGDTSHR
SCHEMBL3630867 0.70 NOS3 (0.45) PARP1ALDH1A1L3MBTL1HPGDTSHR
SCHEMBL2480404 0.68 PARP1 (0.56) PARP1ALDH1A1L3MBTL1CD44HSD17B10
SCHEMBL20364104 0.67 ALDH1A1 (0.48) PARP1ALDH1A1L3MBTL1CD44HSD17B10
SCHEMBL6751983 0.65 PARP1 (0.44) PARP1ALDH1A1L3MBTL1CD44HSD17B10
SCHEMBL2768935 0.65 PARP1 (0.53) PARP1ALDH1A1L3MBTL1HSD17B10TSHR
SCHEMBL12657972 0.65 PARP1 (0.44) PARP1ALDH1A1L3MBTL1CD44HSD17B10
SCHEMBL192953 0.65 CD44 (0.38) PARP1ALDH1A1CD44HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6706924-B2 INCLUDES A STEP IN WHICH ORTHO-NITROTOLUENE IS REACTED WITH ONE OR MORE ACRYLIC ACID DERIVATIVES SUCH AS ACRYLONITRILE BAYER AKTIENGESELLSCHAFT (DE) 2004-03-16 US claimed
EP-1345888-A1 METHOD FOR THE PRODUCTION OF 1,5-NAPHTHALENEDIAMINE Bayer Aktiengesellschaft (DE) 2003-09-24 EP claimed
US-20020103401-A1 Process for the production of 1,5-naphthalenediamine BAYER AKTIENGESELLSCHAFT (DE) 2002-08-01 US claimed
WO-2002051792-A1 METHOD FOR THE PRODUCTION OF 1,5-NAPHTHALENEDIAMINE BAYER AKTIENGESELLSCHAFT (DE) 2002-07-04 WO claimed
US-6706924-B2 INCLUDES A STEP IN WHICH ORTHO-NITROTOLUENE IS REACTED WITH ONE OR MORE ACRYLIC ACID DERIVATIVES SUCH AS ACRYLONITRILE BAYER AKTIENGESELLSCHAFT (DE) 2004-03-16 US disclosed
EP-1345888-A1 METHOD FOR THE PRODUCTION OF 1,5-NAPHTHALENEDIAMINE Bayer Aktiengesellschaft (DE) 2003-09-24 EP disclosed
US-20020103401-A1 Process for the production of 1,5-naphthalenediamine BAYER AKTIENGESELLSCHAFT (DE) 2002-08-01 US disclosed
WO-2002051792-A1 METHOD FOR THE PRODUCTION OF 1,5-NAPHTHALENEDIAMINE BAYER AKTIENGESELLSCHAFT (DE) 2002-07-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020103401-A1 Process for the production of 1,5-naphthalenediamine BBOX1, CYP4B1, NAT1 PARP1 1388/4885ALDH1A1 455/4885L3MBTL1 4585/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.