SCHEMBL6755686

SCHEMBL6755686

CC(C)([CH]C(=O)c1ccc(S(C)(=O)=O)cc1)C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.44
AKR1C3 P42330 2/20 0.44
PTGS2 P35354 6/20 0.41
EPHX2 P34913 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
ENPP2 Q13822 1/20 0.41
GSR P00390 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6759432 0.81 ALDH5A1 (0.47) MAOB
SCHEMBL1381443 0.74 CA2 (0.65) AKR1C3PTGS2ENPP2GSR
SCHEMBL6656686 0.73 GSR (0.51) AKR1C3EPHX2NR1H4ENPP2GSR
Hydrochloric Acid SCHEMBL14482763 0.72 CA2 (0.63) AKR1C3PTGS2ENPP2GSR
SCHEMBL3056916 0.72 AKR1C3 (0.53) MAOBAKR1C3PTGS2ENPP2GSR
SCHEMBL14754379 0.72 AKR1C3 (0.49) MAOBAKR1C3PTGS2ENPP2GSR
SCHEMBL13543239 0.71 ENPP2 (0.50) MAOBAKR1C3PTGS2EPHX2NR1H4
SCHEMBL27470345 0.71 TGM2 (0.58) MAOBAKR1C3PTGS2ENPP2GSR
SCHEMBL4321082 0.69 ENPP2 (0.58) AKR1C3PTGS2ENPP2GSR
SCHEMBL29356248 0.69 CA2 (0.69) PTGS2ENPP2GSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716878-B1 BACTERICIDE, ANTIPROTOZOAL; VANCOMYCIN RESISTANT ENTEROCOCCI AND BETA-LACTAM ANTIBIOTIC-RESISTANT BACTERIA, METHICILLIN-RESISTANT STAPHYLOCOCCUS AUREUS; HYDROXAMIC ACID AND N-FORMYL SUBTITUTED ALKYLAMIDES VERNALIS (OXFORD) LIMITED (GB) 2004-04-06 US claimed
US-6716878-B1 BACTERICIDE, ANTIPROTOZOAL; VANCOMYCIN RESISTANT ENTEROCOCCI AND BETA-LACTAM ANTIBIOTIC-RESISTANT BACTERIA, METHICILLIN-RESISTANT STAPHYLOCOCCUS AUREUS; HYDROXAMIC ACID AND N-FORMYL SUBTITUTED ALKYLAMIDES VERNALIS (OXFORD) LIMITED (GB) 2004-04-06 US disclosed