SCHEMBL6762069

SCHEMBL6762069

CS(=O)(=O)c1ccc(CN2Cc3ccc(C(=O)O)cc3C2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA4 P22748 2/20 0.49
CA9 Q16790 2/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PTGS1 P23219 1/20 0.46
HDAC1 Q13547 6/20 0.44
HDAC4 P56524 4/20 0.44
HDAC6 Q9UBN7 4/20 0.44
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.41
ENPP2 Q13822 1/20 0.41
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
ERCC5 P28715 1/20 0.40
FEN1 P39748 1/20 0.40
TAS2R14 Q9NYV8 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
PRMT5 O14744 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6767486 0.84 MEN1 (0.49) CA1CA2CA4CA9MEN1
SCHEMBL2065219 0.84 HDAC1 (0.59) MEN1KMT2AHDAC1HDAC4HDAC6
SCHEMBL12446495 0.84 HDAC1 (0.49) MEN1KMT2AHDAC1HDAC4HDAC6
SCHEMBL7984900 0.82 L3MBTL1 (0.53) CA1CA2MEN1KMT2AHDAC1
SCHEMBL12446493 0.80 HDAC1 (0.52) MEN1KMT2AHDAC1HDAC4HDAC6
SCHEMBL6704915 0.79 ERCC5 (0.44) CA1CA2CA4CA9PTGS1
SCHEMBL6764235 0.78 MAPK1 (0.48) MEN1KMT2AHDAC1HDAC4HDAC6
SCHEMBL6765162 0.78 CA1 (0.77) CA1CA2CA4CA9MEN1
SCHEMBL8344881 0.77 RORC (0.43) ITGB3ITGA2B
SCHEMBL12363333 0.77 KMT2A (0.47) CA1CA9MEN1KMT2AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040038973-A1 Treating osteoarthritis or rheumatoid arthritis NAHRA JOE (US) 2004-02-26 US claimed
WO-2004014365-A1 PHTHALIMIDE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed
US-20040038973-A1 Treating osteoarthritis or rheumatoid arthritis NAHRA JOE (US) 2004-02-26 US disclosed
WO-2004014365-A1 PHTHALIMIDE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040038973-A1 Treating osteoarthritis or rheumatoid arthritis MMP13, MMP11, MMP9 CA1 724/4885CA2 300/4885CA4 591/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.