SCHEMBL6763168

SCHEMBL6763168

Cc1ccc2oc(-c3ccc(O)c(C)c3)nc(=O)c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
CSNK2A2 P19784 7/20 0.45
CSNK2B P67870 7/20 0.45
CSNK2A1 P68400 7/20 0.45
KDM4E B2RXH2 4/20 0.44
TP53 P04637 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HSD17B10 Q99714 2/20 0.44
MAPT P10636 4/20 0.43
SNCA P37840 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
NQO1 P15559 1/20 0.41
PKM P14618 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6763157 0.82 CSNK2A2 (0.50) NPC1RAB9ACSNK2A2CSNK2BCSNK2A1
SCHEMBL17254780 0.81 MAOB (0.46) NPC1RAB9AKDM4ETP53ALDH1A1
SCHEMBL9608562 0.76 RAB9A (0.68) NPC1RAB9AKDM4ETP53ALDH1A1
SCHEMBL11320611 0.73 NPC1 (0.59) NPC1RAB9AKDM4ETP53ALDH1A1
SCHEMBL311433 0.73 ALOX5 (0.58) NPC1RAB9AKDM4ETP53ALDH1A1
SCHEMBL9608577 0.73 GPR119 (0.52) NPC1RAB9AKDM4ETP53ALDH1A1
SCHEMBL17254783 0.73 MAOB (0.59) NPC1RAB9ACSNK2A2CSNK2BCSNK2A1
SCHEMBL311263 0.73 ESR1 (0.61) NPC1RAB9ACSNK2A2CSNK2BCSNK2A1
SCHEMBL7600946 0.72 ELANE (0.54) NPC1RAB9ACSNK2A2CSNK2BCSNK2A1
SCHEMBL5307439 0.71 NPC1 (0.60) NPC1RAB9AKDM4ETP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723742-B2 TREATMENT OF DISEASES WHICH CAUSE EXCESS OF IRON IN HUMAN OR ANIMAL BODY OR ARE CAUSED BY IT NOVARTIS AG. (CH) 2004-04-20 US disclosed
US-20030203954-A1 Substituted 3, 5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators LATTMANN RENE (CH) 2003-10-30 US disclosed
US-6596750-B2 Compounds have useful pharmaceutical properties and are particularly active as iron chelators. They can be used for the treatment of iron overload in warm-blooded animals. NOVARTIS AG (CH) 2003-07-22 US disclosed
US-20030069273-A1 Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators LATTMANN RENE (CH) 2003-04-10 US disclosed
EP-0914118-B1 SUBSTITUTED 3,5-DIPHENYL-1,2,4-TRIAZOLES AND THEIR USE AS PHARMACEUTICAL METAL CHELATORS NOVARTIS AG (CH) 2002-10-23 EP disclosed
US-6465504-B1 Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators NOVARTIS AG (CH) 2002-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030069273-A1 Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators TFRC, SLC40A1, FECH NPC1 2448/4885RAB9A 2542/4885CSNK2A2 4369/4885
US-20030203954-A1 Substituted 3, 5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators TFRC, SLC40A1, FECH NPC1 2448/4885RAB9A 2542/4885CSNK2A2 4369/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.