SCHEMBL6763508

SCHEMBL6763508

O=C1COC(c2ccccc2OCCN2CCCCC2)=NN1c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
CYP2D6 P10635 1/20 0.47
ALDH1A1 P00352 5/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
PKM P14618 1/20 0.46
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.44
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HRH1 P35367 2/20 0.44
DRD2 P14416 2/20 0.44
DRD1 P21728 2/20 0.44
DRD3 P35462 2/20 0.44
DRD4 P21917 1/20 0.44
DRD5 P21918 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6763534 0.99 KDM4E (0.50) KDM4ESMN1; SMN2CYP2D6ALDH1A1KMT2A
SCHEMBL6766532 0.95 KDM4E (0.53) KDM4ESMN1; SMN2CYP2D6ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL6773276 0.94 KDM4E (0.52) KDM4ESMN1; SMN2CYP2D6ALDH1A1KMT2A
SCHEMBL5779094 0.91 KDM4E (0.54) KDM4ESMN1; SMN2ALDH1A1POLBL3MBTL1
Hydrochloric Acid SCHEMBL6768032 0.90 KDM4E (0.53) KDM4EALDH1A1LMNAPOLBHTT
SCHEMBL6763407 0.87 TSHR (0.42) KDM4ESMN1; SMN2CYP2D6KMT2AMEN1
Hydrochloric Acid SCHEMBL6766958 0.86 TSHR (0.41) KDM4ESMN1; SMN2CYP2D6KMT2AMEN1
SCHEMBL6768461 0.86 TDP1 (0.41) KDM4ESMN1; SMN2CYP2D6KMT2AMEN1
Hydrochloric Acid SCHEMBL6766915 0.85 TDP1 (0.40) KDM4ESMN1; SMN2CYP2D6KMT2AMEN1
SCHEMBL5780359 0.84 KDM4E (0.49) KDM4EPOLBL3MBTL1DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825192-B1 NON-N-METHYL-D-ASPARTATE (NON- NMDA) EXCITATORY AMINO ACID RECEPTOR ANTAGONISTIC ACTION, FOR EXAMPLE 2-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) RECEPTOR ANTAGONISTIC ACTION EISAI CO., LTD. (JP) 2004-11-30 US disclosed
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP disclosed