SCHEMBL6766532

SCHEMBL6766532

O=C1COC(c2ccccc2OCCCN2CCCCC2)=NN1c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.53
ALDH1A1 P00352 6/20 0.53
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
PKM P14618 1/20 0.53
CYP2D6 P10635 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.51
HTT P42858 1/20 0.51
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
POLB P06746 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.46
HRH1 P35367 2/20 0.45
HRH3 Q9Y5N1 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C19 P33261 1/20 0.44
USP2 O75604 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6773276 0.99 KDM4E (0.52) KDM4EALDH1A1KMT2AMEN1PKM
SCHEMBL6763508 0.95 KDM4E (0.52) KDM4EALDH1A1KMT2AMEN1PKM
SCHEMBL6763534 0.94 KDM4E (0.50) KDM4EALDH1A1KMT2AMEN1PKM
SCHEMBL5779094 0.86 KDM4E (0.54) KDM4EALDH1A1L3MBTL1POLBSMN1; SMN2
Hydrochloric Acid SCHEMBL6768032 0.85 KDM4E (0.53) KDM4EALDH1A1L3MBTL1HTTLMNA
SCHEMBL6763407 0.82 TSHR (0.42) KDM4EKMT2AMEN1CYP2D6SMN1; SMN2
SCHEMBL5779725 0.81 KDM4E (0.44) KDM4EALDH1A1SMN1; SMN2HRH1
Hydrochloric Acid SCHEMBL6766958 0.81 TSHR (0.41) KDM4EKMT2AMEN1CYP2D6SMN1; SMN2
SCHEMBL6768461 0.81 TDP1 (0.41) KDM4EKMT2AMEN1CYP2D6SMN1; SMN2
Hydrochloric Acid SCHEMBL5779062 0.80 KDM4E (0.43) KDM4EALDH1A1SMN1; SMN2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP claimed
US-6825192-B1 NON-N-METHYL-D-ASPARTATE (NON- NMDA) EXCITATORY AMINO ACID RECEPTOR ANTAGONISTIC ACTION, FOR EXAMPLE 2-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) RECEPTOR ANTAGONISTIC ACTION EISAI CO., LTD. (JP) 2004-11-30 US disclosed
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP disclosed