SCHEMBL6768461

SCHEMBL6768461

O=C1COC(c2ncccc2OCCN2CCCC2)=NN1c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
DRD1 P21728 4/20 0.41
DRD3 P35462 3/20 0.41
DRD2 P14416 3/20 0.41
HRH1 P35367 3/20 0.41
DRD4 P21917 2/20 0.41
DRD5 P21918 2/20 0.41
TSHR P16473 1/20 0.40
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
CYP2D6 P10635 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6766915 0.99 TDP1 (0.40) TDP1DRD1DRD3DRD2HRH1
SCHEMBL6763407 0.99 TSHR (0.42) TDP1DRD1DRD3DRD2HRH1
Hydrochloric Acid SCHEMBL6766958 0.98 TSHR (0.41) TDP1DRD1DRD3DRD2HRH1
SCHEMBL5779879 0.92 POLB (0.45) DRD1DRD4DRD5KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL5777092 0.91 POLB (0.44) DRD1DRD4DRD5KDM4EMEN1
SCHEMBL6763534 0.87 KDM4E (0.50) TDP1DRD1DRD3DRD2HRH1
SCHEMBL6763508 0.86 KDM4E (0.52) TDP1DRD1DRD3DRD2HRH1
SCHEMBL6763485 0.85 CYP11B1 (0.36) TDP1DRD3TSHRKDM4ESMN1; SMN2
SCHEMBL6767694 0.83 CHRNB4 (0.41) DRD1DRD3DRD2HRH1TSHR
SCHEMBL5781776 0.83 HTR7 (0.38) TDP1DRD1DRD3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP claimed
US-6825192-B1 NON-N-METHYL-D-ASPARTATE (NON- NMDA) EXCITATORY AMINO ACID RECEPTOR ANTAGONISTIC ACTION, FOR EXAMPLE 2-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) RECEPTOR ANTAGONISTIC ACTION EISAI CO., LTD. (JP) 2004-11-30 US disclosed
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP disclosed