SCHEMBL6763545

SCHEMBL6763545

O=C1C(c2ccccc2)OC(c2ccccc2)=NN1c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
GFER P55789 1/20 0.48
CES2 O00748 13/20 0.44
LOX P28300 1/20 0.43
LOXL3 P58215 1/20 0.43
LOXL4 Q96JB6 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
MAOB P27338 2/20 0.40
CA2 P00918 1/20 0.39
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.37
SLC6A3 Q01959 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28494246 0.67 MAOA (0.61) ALDH1A1CA2LMNARAB9ASLC6A3
SCHEMBL6768350 0.67 KMT2A (0.47) ALDH1A1CES2LOXMAOBCA2
SCHEMBL6766023 0.67 CA2 (0.50) ALDH1A1GFERMAOBCA2LMNA
SCHEMBL8930590 0.65 CES2 (0.65) ALDH1A1GFERCES2LOXLOXL3
SCHEMBL30641875 0.65 ALDH1A1 (1.00) ALDH1A1GFERCES2LOXLOXL3
SCHEMBL6773284 0.65 SMN1; SMN2 (0.44) ALDH1A1GFERCES2LOXLOXL3
SCHEMBL30641876 0.62 ALDH1A1 (0.67) ALDH1A1GFERCES2LOXLOXL3
SCHEMBL17290527 0.62 CES2 (0.57) CES2LOXLOXL3LOXL4LOXL2
SCHEMBL17454853 0.62 MAOB (0.48) ALDH1A1MAOBRAB9A
SCHEMBL28185949 0.62 MAOB (0.48) ALDH1A1MAOBHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825192-B1 NON-N-METHYL-D-ASPARTATE (NON- NMDA) EXCITATORY AMINO ACID RECEPTOR ANTAGONISTIC ACTION, FOR EXAMPLE 2-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) RECEPTOR ANTAGONISTIC ACTION EISAI CO., LTD. (JP) 2004-11-30 US disclosed
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP disclosed