SCHEMBL6763992

SCHEMBL6763992

O=C(O)CNC(=O)CNCS(=O)(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.47
KMT2A Q03164 2/20 0.41
GAA P10253 1/20 0.41
SHMT1 P34896 1/20 0.39
SHMT2 P34897 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
CA1 P00915 7/20 0.38
CA2 P00918 7/20 0.38
ITGAV P06756 1/20 0.37
AKR1B1 P15121 1/20 0.37
USP5 P45974 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6884908 0.85 POLB (0.44) POLBKMT2ASHMT1SHMT2ALDH1A1
SCHEMBL6764149 0.84 ALDH1A1 (0.43) POLBKMT2AALDH1A1CA1CA2
SCHEMBL11888774 0.80 GAA (0.41) POLBKMT2AGAACA1CA2
SCHEMBL6762826 0.77 SHMT1 (0.44) SHMT1SHMT2ALDH1A1TSHRCA1
SCHEMBL6763197 0.75 WDR5 (0.40) POLBCA1CA2USP5
SCHEMBL5124231 0.74 FABP4 (0.46) POLBKMT2AGAAALDH1A1
SCHEMBL493617 0.72 KMT2A (0.42) POLBKMT2AGAAALDH1A1AKR1B1
SCHEMBL6763996 0.72 POLB (0.45) POLBKMT2AGAAALDH1A1
SCHEMBL5115187 0.71 KMT2A (0.41) POLBKMT2AGAAALDH1A1ITGAV
SCHEMBL5115190 0.71 KMT2A (0.41) POLBKMT2AGAAALDH1A1ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040063725-A1 Novel n(phenylsulphonyl)glycine derivatives and their therapeutic use LABORATORIES FOURNIER S.A. (FR) 2004-04-01 US disclosed
EP-1351928-A2 NOVEL N(PHENYLSULPHONYL)GLYCINE DERIVATIVES AND THEIR THERAPEUTIC USE LABORATOIRES FOURNIER S.A. (FR) 2003-10-15 EP disclosed
WO-2002053516-A2 N(PHENYLSULPHONYL)GLYCINE DERIVATIVES AND THEIR THERAPEUTIC USE LABORATOIRES FOURNIER SA (FR) 2002-07-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063725-A1 Novel n(phenylsulphonyl)glycine derivatives and their therapeutic use GLS, GLS2, GLRB POLB 2689/4885KMT2A 3854/4885GAA 492/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.