SCHEMBL6770288

SCHEMBL6770288

CC(C)c1ccc(-n2nc(-c3cccs3)c3c2C(C#N)C(C)(C)CC3=O)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.37
HSD17B10 Q99714 5/20 0.37
ALDH1A1 P00352 4/20 0.37
HPGD P15428 3/20 0.37
ALPL P05186 1/20 0.37
CCNA2 P20248 4/20 0.37
CDK2 P24941 4/20 0.37
POLB P06746 1/20 0.36
MAPT P10636 5/20 0.34
USP2 O75604 3/20 0.34
TSHR P16473 2/20 0.34
CASP1 P29466 2/20 0.34
RXFP1 Q9HBX9 2/20 0.34
CASP7 P55210 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SRC P12931 1/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
LMNA P02545 3/20 0.33
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6767179 0.86 POLB (0.35) KDM4EHSD17B10ALDH1A1HPGDALPL
SCHEMBL6772430 0.85 CCNA2 (0.44) KDM4EALDH1A1HPGDCCNA2CDK2
SCHEMBL6770739 0.85 CCNA2 (0.45) ALDH1A1CCNA2CDK2SRCMEN1
SCHEMBL6766539 0.83 CCNA2 (0.35) CCNA2CDK2SRCMEN1KMT2A
SCHEMBL6776854 0.82 PTGS1 (0.42) KDM4EHSD17B10ALDH1A1HPGDCCNA2
SCHEMBL6775773 0.81 CCNA2 (0.39) ALDH1A1CCNA2CDK2MAPTMEN1
SCHEMBL6771336 0.81 CCNA2 (0.37) CCNA2CDK2SRCMEN1KMT2A
SCHEMBL6767158 0.80 CCNA2 (0.37) CCNA2CDK2MEN1KMT2ALMNA
SCHEMBL6772549 0.80 CCNA2 (0.35) KDM4EALDH1A1CCNA2CDK2MAPT
SCHEMBL7534112 0.79 OPRM1 (0.50) KDM4EHSD17B10ALDH1A1HPGDALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed