SCHEMBL6770960

SCHEMBL6770960

CC(C)c1ccc(-n2nc(C3CC3)c3c2CCCC3=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 4/20 0.43
OPRM1 P35372 3/20 0.39
GRIA2 P42262 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPT P10636 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 2/20 0.36
PKM P14618 2/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CSNK2B P67870 2/20 0.34
CSNK2A1 P68400 2/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
MGLL Q99685 1/20 0.34
CSNK2A2 P19784 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6771990 0.84 OPRM1 (0.54) SRCOPRM1GRIA2CYP1A2CYP2C9
SCHEMBL6767135 0.83 OPRM1 (0.41) SRCOPRM1GRIA2CYP1A2CYP2C9
SCHEMBL6771178 0.83 SRC (0.43) SRCOPRM1GRIA2ALDH1A1PKM
SCHEMBL6166055 0.83 ALDH1A1 (0.46) SRCOPRM1MAPTALDH1A1PKM
SCHEMBL6777334 0.81 L3MBTL1 (0.47) OPRM1GRIA2CYP1A2CYP2C9MAPT
SCHEMBL6770500 0.81 OPRM1 (0.61) SRCOPRM1
SCHEMBL6769850 0.81 OPRM1 (0.38) OPRM1GRIA2CYP1A2CYP2C9MAPT
SCHEMBL6770454 0.78 ALDH1A1 (0.48) SRCOPRM1GRIA2CYP1A2CYP2C9
SCHEMBL6771814 0.78 SRC (0.60) SRCOPRM1MAPTALDH1A1KDM4E
SCHEMBL6772956 0.75 SRC (0.49) SRCOPRM1MAPTL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed