SCHEMBL6771990

SCHEMBL6771990

Cc1nn(-c2ccc(C(C)C)cc2)c2c1C(=O)CCC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.54
HTT P42858 1/20 0.45
SRC P12931 3/20 0.43
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
GRIA2 P42262 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
MGLL Q99685 1/20 0.37
MAPT P10636 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6767135 0.88 OPRM1 (0.41) OPRM1HTTSRCLMNAALDH1A1
SCHEMBL6770960 0.84 SRC (0.43) OPRM1HTTSRCLMNAALDH1A1
SCHEMBL6770286 0.83 OPRM1 (0.56) OPRM1HTTSRCALDH1A1PKM
SCHEMBL6162529 0.82 OPRM1 (0.56) OPRM1HTTSRCLMNAALDH1A1
SCHEMBL6770454 0.82 ALDH1A1 (0.48) OPRM1HTTSRCLMNAALDH1A1
SCHEMBL6771511 0.80 L3MBTL1 (0.49) OPRM1HTTLMNAALDH1A1PKM
SCHEMBL6770401 0.80 OPRM1 (0.77) OPRM1HTTLMNAALDH1A1NPSR1
SCHEMBL6770476 0.79 OPRM1 (0.45) OPRM1LMNAALDH1A1PKMSMN1; SMN2
SCHEMBL6769828 0.77 OPRM1 (0.67) OPRM1HTTSRCLMNAALDH1A1
SCHEMBL6767074 0.76 OPRM1 (0.41) OPRM1HTTSRCLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed