SCHEMBL6771042

SCHEMBL6771042

CCCc1nn(-c2cccc(Cl)c2)c2c1C(=O)CC(C)C2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 1/20 0.40
SRC P12931 1/20 0.40
GAA P10253 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SLC5A1 P13866 2/20 0.38
MEN1 O00255 1/20 0.37
HSP90AA1 P07900 1/20 0.37
KMT2A Q03164 1/20 0.37
CSNK2A2 P19784 2/20 0.36
CSNK2B P67870 2/20 0.36
CSNK2A1 P68400 2/20 0.36
ABCG2 Q9UNQ0 2/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
KCNH2 Q12809 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6164477 0.87 ABCG2 (0.43) ALDH1A1LMNAMAPTNPSR1KMT2A
SCHEMBL6770490 0.86 ALDH1A1 (0.42) ALDH1A1LMNAMAPTSRCGAA
SCHEMBL6769517 0.86 SRC (0.39) ALDH1A1LMNASRCMEN1HSP90AA1
SCHEMBL6777711 0.82 OPRM1 (0.45) ALDH1A1LMNAMAPTSRCGAA
SCHEMBL6771081 0.82 ALDH1A1 (0.58) ALDH1A1LMNAMAPTSRCGAA
SCHEMBL6767198 0.81 L3MBTL1 (0.44) ALDH1A1LMNAMAPTGAANPSR1
SCHEMBL6770294 0.81 SRC (0.36) ALDH1A1LMNASRCSLC5A1CSNK2A2
SCHEMBL6771222 0.81 OPRM1 (0.47) ALDH1A1MAPTSRCMEN1KMT2A
SCHEMBL6772480 0.80 ALDH1A1 (0.67) ALDH1A1LMNASRCGAANPSR1
SCHEMBL6770768 0.80 SRC (0.41) ALDH1A1LMNAMAPTSRCGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed