SCHEMBL6772323

SCHEMBL6772323

COc1cccc(-n2nc(C3CC3)c3c2CC(C)CC3=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.41
NSD2 O96028 1/20 0.39
NSD1 Q96L73 1/20 0.39
NSD3 Q9BZ95 1/20 0.39
LPAR5 Q9H1C0 1/20 0.39
HPSE Q9Y251 1/20 0.39
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
RAB9A P51151 3/20 0.38
KMT2A Q03164 3/20 0.38
MAPT P10636 2/20 0.38
HTT P42858 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
SRC P12931 1/20 0.38
MGLL Q99685 1/20 0.37
OPRM1 P35372 1/20 0.37
S1PR4 O95977 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6772063 0.87 OPRM1 (0.48) SMN1; SMN2RAB9AKMT2AMAPTHTT
SCHEMBL6771222 0.86 OPRM1 (0.47) SMN1; SMN2KMT2AMAPTL3MBTL1MEN1
SCHEMBL6770575 0.86 GPBAR1 (0.39) GPBAR1NSD2NSD1NSD3LPAR5
SCHEMBL6168193 0.84 ABCG2 (0.42) HPGDSMN1; SMN2RAB9AKMT2AMAPT
SCHEMBL6775862 0.83 ABCG2 (0.39) HPGDSMN1; SMN2RAB9AKMT2AMAPT
SCHEMBL6766708 0.83 RIPK2 (0.48) HPGDSMN1; SMN2RAB9AKMT2AMAPT
SCHEMBL6772956 0.83 SRC (0.49) GPBAR1NSD2NSD1NSD3LPAR5
SCHEMBL6766537 0.81 ALDH1A1 (0.41) HPGDSMN1; SMN2RAB9AKMT2AMAPT
SCHEMBL6771516 0.81 OPRM1 (0.58) SRCOPRM1
SCHEMBL6771827 0.81 ABCG2 (0.37) HPGDSMN1; SMN2RAB9AKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed