SCHEMBL6772063

SCHEMBL6772063

COc1cccc(-n2nc(C)c3c2CC(C)CC3=O)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.48
SRC P12931 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 1/20 0.40
MGLL Q99685 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
MAP4K4 O95819 1/20 0.39
AURKB Q96GD4 1/20 0.39
SRPK1 Q96SB4 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6772323 0.87 GPBAR1 (0.41) OPRM1SRCSMN1; SMN2RAB9ANPC1
SCHEMBL6777711 0.86 OPRM1 (0.45) OPRM1SRCSMN1; SMN2MEN1KMT2A
SCHEMBL6775862 0.86 ABCG2 (0.39) SRCSMN1; SMN2RAB9ANPC1MEN1
SCHEMBL6766708 0.86 RIPK2 (0.48) OPRM1SRCSMN1; SMN2RAB9ANPC1
SCHEMBL6770505 0.85 OPRM1 (0.46) OPRM1SRCSMN1; SMN2RAB9ANPC1
SCHEMBL6167870 0.84 ALDH1A1 (0.49) OPRM1SMN1; SMN2RAB9ANPC1MEN1
SCHEMBL6766537 0.84 ALDH1A1 (0.41) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL6771827 0.83 ABCG2 (0.37) SRCSMN1; SMN2RAB9ANPC1MEN1
SCHEMBL6770366 0.81 SRC (0.56) OPRM1SRCSMN1; SMN2RAB9ANPC1
SCHEMBL6772144 0.79 RIPK2 (0.36) SRCSMN1; SMN2RAB9ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed