SCHEMBL6777392

SCHEMBL6777392

CC(C)C1CC(=O)c2c(C(C)(C)C)nn(-c3ccc(I)cc3)c2C1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.36
GRIA2 P42262 4/20 0.30
CYP1A2 P05177 3/20 0.30
CYP2C9 P11712 2/20 0.30
BUB1 O43683 1/20 0.30
CYP2D6 P10635 1/20 0.30
HSP90AB1 P08238 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7490727 0.88 L3MBTL1 (0.36) DHODHGRIA2CYP1A2CYP2C9CYP2D6
SCHEMBL6164978 0.88 DHODH (0.41) DHODHBUB1
SCHEMBL6771481 0.84 OPRM1 (0.43) DHODHBUB1HSP90AB1
SCHEMBL6771234 0.84 CSNK2A2 (0.35) BUB1
SCHEMBL6769804 0.83 PPARA (0.38) DHODHBUB1
SCHEMBL6770489 0.83 DHODH (0.35) DHODHBUB1
SCHEMBL6776388 0.82 OPRM1 (0.38) DHODHBUB1
SCHEMBL6771327 0.82 DHODH (0.32) DHODH
SCHEMBL6770539 0.81 SRC (0.39) DHODH
SCHEMBL6767248 0.80 DHODH (0.35) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed