SCHEMBL6778077

SCHEMBL6778077

COc1ccc(CCC(Cc2ccc(OC)c(OC)c2)CN2C[C@H]3CC[C@@H](C2=O)N3Cc2ccccc2)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.44
KMT2A Q03164 1/20 0.42
POLB P06746 3/20 0.41
MAPK1 P28482 2/20 0.41
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 2/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6780165 0.95 SIGMAR1 (0.46) SIGMAR1POLBMAPK1PDE4APDE4B
SCHEMBL6784175 0.90 SIGMAR1 (0.45) SIGMAR1POLBMAPK1PDE4APDE4B
SCHEMBL6779144 0.86 SIGMAR1 (0.50) SIGMAR1POLBMAPK1PDE4APDE4B
SCHEMBL6784327 0.83 SIGMAR1 (0.47) SIGMAR1POLBMAPK1PDE4APDE4B
SCHEMBL6774415 0.82 BCHE (0.39) SIGMAR1KMT2AALDH1A1MAPT
SCHEMBL6779167 0.78 SIGMAR1 (0.46) SIGMAR1POLBMAPK1PDE4APDE4B
SCHEMBL6779579 0.77 BCHE (0.42) SIGMAR1KMT2AALDH1A1TSHRMAPT
SCHEMBL6784683 0.75 OPRM1 (0.41) SIGMAR1ALDH1A1
SCHEMBL6776517 0.73 FKBP5 (0.45) SIGMAR1KMT2APOLBMAPK1PDE4A
SCHEMBL6775893 0.69 OPRM1 (0.49) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818643-B1 3,9-DIAZABICYCLO(3.3.1)NONAN-2-ONE DERIVATIVES; PEPTIDYL-PROLYL ISOMERASE (PPIASE OR ROTAMASE) INHIBITORS; NEUROPROTECTIVE AGENTS BRISTOL-MYERS SQUIBB COMPANY 2004-11-16 US disclosed