SCHEMBL6776517

SCHEMBL6776517

COc1ccc(CCC(CCc2ccccc2)CN2CC3CCCC(C2=O)N3C(=O)OC(C)(C)C)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FKBP5 Q13451 2/20 0.45
POLB P06746 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42
FKBP1A P62942 4/20 0.40
ALDH1A1 P00352 5/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KMT2A Q03164 1/20 0.40
MAPK1 P28482 1/20 0.40
TSHR P16473 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6780351 0.85 KMT2A (0.40) POLBFKBP1AL3MBTL1KMT2A
SCHEMBL6778877 0.84 FKBP5 (0.51) FKBP5POLBNPC1TP53RAB9A
SCHEMBL6778408 0.83 FKBP5 (0.50) FKBP5POLBNPC1TP53RAB9A
SCHEMBL15436137 0.79 FKBP5 (0.49) FKBP5POLBNPC1TP53RAB9A
SCHEMBL6775961 0.78 KMT2A (0.42) FKBP5POLBFKBP1AL3MBTL1KMT2A
SCHEMBL6780165 0.78 SIGMAR1 (0.46) POLBNPC1TP53RAB9AALDH1A1
SCHEMBL6785002 0.77 KMT2A (0.41) FKBP5POLBFKBP1AL3MBTL1KMT2A
SCHEMBL6778841 0.77 KMT2A (0.41) FKBP5POLBFKBP1AL3MBTL1KMT2A
SCHEMBL6776495 0.76 FKBP5 (0.51) FKBP5FKBP1AKMT2A
SCHEMBL6784892 0.76 FKBP1A (0.48) FKBP5FKBP1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818643-B1 3,9-DIAZABICYCLO(3.3.1)NONAN-2-ONE DERIVATIVES; PEPTIDYL-PROLYL ISOMERASE (PPIASE OR ROTAMASE) INHIBITORS; NEUROPROTECTIVE AGENTS BRISTOL-MYERS SQUIBB COMPANY 2004-11-16 US disclosed