SCHEMBL6785203

SCHEMBL6785203

CC(C)(C)OC(=O)N1CCN(NC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.62
S1PR2 O95136 1/20 0.56
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
CYP2C19 P33261 2/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MAPT P10636 2/20 0.46
PKM P14618 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MMP13 P45452 1/20 0.46
LMNA P02545 2/20 0.46
STS P08842 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581249 0.87 S1PR2 (0.56) CYP2D6S1PR2KMT2AMEN1SMN1; SMN2
SCHEMBL21819487 0.87 KMT2A (0.64) CYP2D6KMT2AMEN1SMN1; SMN2CYP2C19
SCHEMBL21819347 0.85 GPR119 (0.55) CYP2D6S1PR2KMT2AMEN1SMN1; SMN2
SCHEMBL3093877 0.82 MEN1 (0.68) S1PR2KMT2AMEN1
SCHEMBL194951 0.80 CYP2D6 (0.72) CYP2D6SMN1; SMN2CYP2C19HTTMAPT
SCHEMBL4603719 0.80 HDAC4 (0.63) KMT2AMEN1MAPTPKMKDM4E
SCHEMBL5752686 0.79 HTR1A (0.60) KMT2AMEN1
Water SCHEMBL3089403 0.79 CYP2D6 (0.70) CYP2D6SMN1; SMN2CYP2C19HTTMAPT
SCHEMBL21819310 0.78 KMT2A (0.54) S1PR2KMT2AMEN1SMN1; SMN2HTT
SCHEMBL17807228 0.78 MAPT (0.62) S1PR2KMT2AMEN1SMN1; SMN2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed