SCHEMBL679785

SCHEMBL679785

CS(=O)(=O)NC(=O)c1ccc(Oc2cccc(-c3ccccc3)c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 9/20 0.62
BCL2L1 Q07817 7/20 0.62
SCN9A Q15858 2/20 0.52
HDAC8 Q9BY41 1/20 0.50
GALK1 P51570 1/20 0.49
CASP6 P55212 1/20 0.49
PLEC Q15149 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
PGR P06401 1/20 0.48
FFAR1 O14842 1/20 0.48
FFAR4 Q5NUL3 1/20 0.48
SCN3A Q9NY46 1/20 0.47
NR1H4 Q96RI1 1/20 0.47
TRPV1 Q8NER1 1/20 0.46
MMP1 P03956 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL680289 0.90 MCL1 (0.70) MCL1BCL2L1SCN9APGRSCN3A
SCHEMBL680466 0.84 EZH2 (0.54) MCL1BCL2L1SCN9AHDAC8TDP1
SCHEMBL680286 0.84 PGR (0.60) MCL1BCL2L1SCN9APGR
SCHEMBL678831 0.83 BCL2L1 (0.52) MCL1BCL2L1SCN9AHDAC8PGR
SCHEMBL678903 0.83 BCL2L1 (0.52) MCL1BCL2L1SCN9AADORA3PGR
SCHEMBL680849 0.82 PTPN1 (0.52) MCL1BCL2L1SCN9AHDAC8SCN3A
SCHEMBL31331542 0.81 SCN9A (0.64) MCL1BCL2L1SCN9ASCN3A
SCHEMBL679983 0.81 ACACB (0.50) MCL1BCL2L1SCN3A
SCHEMBL679782 0.81 SCN9A (0.50) MCL1BCL2L1SCN9AHDAC8PGR
SCHEMBL679146 0.81 SCN9A (0.52) MCL1BCL2L1SCN9ASCN3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010207-A1 Chemical Compounds SCN1A, SCN1B, SCN7A MCL1 2739/4885BCL2L1 3284/4885SCN9A 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.