SCHEMBL6799012

SCHEMBL6799012

O=C(O)c1cccc(NC(=O)c2ccccc2-c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APOB P04114 5/20 0.66
NR1H4 Q96RI1 4/20 0.63
PPARG P37231 2/20 0.63
PPARD Q03181 2/20 0.63
PPARA Q07869 1/20 0.60
RXFP1 Q9HBX9 2/20 0.59
HTT P42858 2/20 0.58
KCNK3 O14649 2/20 0.57
KCNK9 Q9NPC2 1/20 0.57
MTTP P55157 4/20 0.56
ALDH1A1 P00352 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CHRNB2 P17787 1/20 0.55
CHRNB4 P30926 1/20 0.55
CHRNA3 P32297 1/20 0.55
CHRNA4 P43681 1/20 0.55
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7607266 0.99 APOB (0.65) APOBNR1H4PPARGPPARDPPARA
SCHEMBL7605815 0.93 APOB (0.63) APOBNR1H4PPARGPPARDRXFP1
SCHEMBL7607259 0.89 APOB (0.59) APOBNR1H4PPARGPPARDRXFP1
SCHEMBL7613563 0.89 APOB (0.59) APOBNR1H4PPARGPPARDPPARA
SCHEMBL31393757 0.87 CHRNB2 (0.71) APOBHTTMTTPALDH1A1CHRNB2
SCHEMBL7048961 0.87 CHRNB2 (0.71) NR1H4HTTALDH1A1L3MBTL1CHRNB2
SCHEMBL3726223 0.86 NPC1 (0.61) APOBMTTPALDH1A1CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL7611573 0.86 CHRNB2 (0.69) NR1H4HTTALDH1A1L3MBTL1CHRNB2
SCHEMBL7612180 0.86 MTTP (0.61) APOBNR1H4PPARGPPARDPPARA
SCHEMBL7607240 0.86 APOB (0.61) APOBNR1H4PPARGPPARDRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040058903-A1 Benzamide compounds as apo b secretion inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-03-25 US disclosed
EP-1326835-A1 BENZAMIDE COMPOUNDS AS APO B SECRETION INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-16 EP disclosed
EP-1301464-A1 BIPHENYLCARBOXYLIC ACID AMIDES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 2003-04-16 EP disclosed
WO-2002028835-A1 BENZAMIDE COMPOUNDS AS APO B SECRETION INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-04-11 WO disclosed
US-20020032238-A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-03-14 US disclosed
WO-2002004403-A1 BIPHENYLCARBOXYLIC ACID AMIDES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-01-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020032238-A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments MTTP, CETP, FABP1 APOB 45/4885NR1H4 99/4885PPARG 86/4885
US-20040058903-A1 Benzamide compounds as apo b secretion inhibitors APOB, APOL1, SCARB1 APOB 1/4885NR1H4 245/4885PPARG 899/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.