SCHEMBL6800561

SCHEMBL6800561

CCOC(=O)CC(C)(C)Cc1ccc(OC)cc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 9/20 0.39
HPGD P15428 7/20 0.39
GAA P10253 4/20 0.39
MAPT P10636 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
TSHR P16473 1/20 0.39
KDM4E B2RXH2 5/20 0.38
HSD17B10 Q99714 2/20 0.38
POLB P06746 2/20 0.38
GLA P06280 1/20 0.38
CASP1 P29466 1/20 0.38
NPC1 O15118 4/20 0.38
RAB9A P51151 3/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806054 0.85 CA12 (0.39) SMN1; SMN2ALDH1A1HPGDCYP1A2CYP2D6
SCHEMBL13742193 0.80 PPARG (0.47) SMN1; SMN2ALDH1A1HPGDGAAMAPT
SCHEMBL6809494 0.79 KMT2A (0.48) SMN1; SMN2ALDH1A1HPGDGAAMAPT
SCHEMBL6809156 0.78 ITGB3 (0.44) L3MBTL1
SCHEMBL432804 0.78 CYP4F2 (0.50) ALDH1A1HPGDGAAMAPTCYP1A2
SCHEMBL4508144 0.77 CYP4F2 (0.49) SMN1; SMN2ALDH1A1HPGDGAACYP1A2
SCHEMBL6803826 0.76 ALDH1A1 (0.39) SMN1; SMN2ALDH1A1GAAMAPTCYP1A2
SCHEMBL6809490 0.74 MEN1 (0.43) SMN1; SMN2ALDH1A1HPGDGAAMAPT
SCHEMBL7352155 0.74 HSD17B10 (0.48) SMN1; SMN2ALDH1A1HPGDGAACYP1A2
SCHEMBL6802346 0.73 APLNR (0.38) ALDH1A1HPGDHSD17B10POLBMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040043994-A1 Gem-substituted alpha v beta 3 antagonists PHARMACIA CORPORATION 2004-03-04 US disclosed
EP-1313705-A1 GEM-SUBSTITUTED ALPHA V BETA 3 INTEGRIN ANTAGONISTS Pharmacia Corporation (US) 2003-05-28 EP disclosed
US-6531494-B1 Gem-substituted αvβ3 antagonists PHARMACIA CORPORATION 2003-03-11 US disclosed
WO-2002018340-A1 GEM-SUBSTITUTED α v β 3 INTEGRIN ANTAGONISTS PHARMACIA CORPORATION (US) 2002-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040043994-A1 Gem-substituted alpha v beta 3 antagonists CACNG5, ITGAV, ITGA5 SMN1; SMN2 1777/4885ALDH1A1 2319/4885HPGD 3958/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.