SCHEMBL6800842

SCHEMBL6800842

C=C(Cc1ccc2c(c1)OCO2)C(=O)N[C@@H](C)C(=O)OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.61
ALDH1A1 P00352 3/20 0.50
RAB9A P51151 3/20 0.50
NPC1 O15118 2/20 0.50
TSHR P16473 2/20 0.50
TP53 P04637 1/20 0.50
MAPT P10636 1/20 0.50
ATM Q13315 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CYP3A4 P08684 2/20 0.49
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
HPGD P15428 1/20 0.47
HRH4 Q9H3N8 1/20 0.47
EDNRA P25101 3/20 0.46
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938275 0.85 CYP3A4 (0.52) ALDH1A1RAB9ANPC1TSHRSMN1; SMN2
SCHEMBL8181400 0.81 ALDH1A1 (0.56) ACEALDH1A1RAB9ANPC1TSHR
SCHEMBL20022971 0.77 ALDH1A1 (0.63) ACEALDH1A1RAB9ANPC1TSHR
Fasidotrilat SCHEMBL29595981 0.76 ACE (1.00) ACEALDH1A1RAB9ANPC1TSHR
SCHEMBL8805246 0.76 MAOB (0.61) ACEALDH1A1RAB9ANPC1MAPT
SCHEMBL8805245 0.76 MAOB (0.61) ACEALDH1A1RAB9ANPC1MAPT
Fasidotril SCHEMBL49006 0.75 ACE (0.88) ACEALDH1A1RAB9ANPC1TSHR
SCHEMBL1650036 0.75 ACE (0.58) ACEALDH1A1RAB9ANPC1TSHR
Fasidotril SCHEMBL7301419 0.75 ACE (0.88) ACEALDH1A1RAB9ANPC1TSHR
SCHEMBL6395296 0.74 MEN1 (0.56) ACEALDH1A1RAB9ANPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6835851-B2 Reacting said alpha - substituted acrylic acid with an chloro acid so as to obtain an acid chloride, now reacting acid chloride thus obtained with an amino ester in presence of an organic base, to acheive coupling BIOPROJET (FR) 2004-12-28 US disclosed
US-20020055645-A1 Process for synthesizing N-(mercaptoacyl) amino acid derivatives from alpha-substituted acrylic acids BIOPROJET (FR) 2002-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020055645-A1 Process for synthesizing N-(mercaptoacyl) amino acid derivatives from alpha-substituted acrylic acids TST, ASS1, SULT1A1 ACE 921/4885ALDH1A1 102/4885RAB9A 2766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.