SCHEMBL6804828

SCHEMBL6804828

COC(=O)CC(C)(C)C(=O)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.57
NR4A2 P43354 2/20 0.56
NR4A1 P22736 1/20 0.56
NR4A3 Q92570 1/20 0.56
PARP10 Q53GL7 1/20 0.54
SRD5A2 P31213 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
NCOR2 Q9Y618 1/20 0.51
ALDH1A1 P00352 3/20 0.50
PPARG P37231 1/20 0.50
PLA2G4B P0C869 1/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3615238 0.87 MAOB (0.55) MAOBNR4A2NR4A1NR4A3PARP10
SCHEMBL5183124 0.83 SRC (0.51) SMN1; SMN2NPC1ALDH1A1KDM4EMEN1
SCHEMBL15189660 0.82 MAOB (0.69) MAOBNR4A2NR4A1NR4A3PARP10
SCHEMBL6399385 0.80 MAPK1 (0.51) PARP10SMN1; SMN2NPC1RAB9AHDAC3
SCHEMBL433676 0.79 MAOB (0.65) MAOBNR4A2NR4A1NR4A3PARP10
SCHEMBL834204 0.78 SMN1; SMN2 (0.61) MAOBNR4A2NR4A1NR4A3PARP10
SCHEMBL10699043 0.78 CA1 (0.48) ALDH1A1KDM4EMAPTADRB2ADRB1
SCHEMBL11809433 0.78 ALDH1A1 (0.56) MAOBNR4A2NR4A1NR4A3PARP10
SCHEMBL978502 0.77 RAB9A (0.71) MAOBNR4A2NR4A1NR4A3PARP10
SCHEMBL810045 0.77 RAB9A (0.63) MAOBNR4A2NR4A1NR4A3PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040043994-A1 Gem-substituted alpha v beta 3 antagonists PHARMACIA CORPORATION 2004-03-04 US disclosed
CN-1471512-A Geminally substituted alphavβ3Integrin antagonists 2004-01-28 CN disclosed
EP-1313705-A1 GEM-SUBSTITUTED ALPHA V BETA 3 INTEGRIN ANTAGONISTS Pharmacia Corporation (US) 2003-05-28 EP disclosed
US-6531494-B1 Gem-substituted αvβ3 antagonists PHARMACIA CORPORATION 2003-03-11 US disclosed
WO-2002018340-A1 GEM-SUBSTITUTED α v β 3 INTEGRIN ANTAGONISTS PHARMACIA CORPORATION (US) 2002-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040043994-A1 Gem-substituted alpha v beta 3 antagonists CACNG5, ITGAV, ITGA5 MAOB 4632/4885NR4A2 2743/4885NR4A1 1826/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.