SCHEMBL6805435

SCHEMBL6805435

CCC(=O)Oc1ccc2c(c1)CC(C)N2C(C)=O

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TNF P01375 5/20 0.53
NOD2 Q9HC29 5/20 0.53
NOD1 Q9Y239 5/20 0.53
NOTUM Q6P988 1/20 0.52
LMNA P02545 1/20 0.51
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
RAB9A P51151 1/20 0.47
PKLR P30613 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6814026 0.85 NOD1 (0.41) TNFNOD2NOD1LMNAMAPT
SCHEMBL2209599 0.82 LMNA (0.68) TNFNOD2NOD1NOTUMLMNA
SCHEMBL2205547 0.82 LMNA (0.68) TNFNOD2NOD1NOTUMLMNA
SCHEMBL12428954 0.82 LMNA (0.68) TNFNOD2NOD1NOTUMLMNA
SCHEMBL26079156 0.78 NOTUM (0.64) TNFNOD2NOD1NOTUMMAPT
SCHEMBL7416927 0.76 NOTUM (0.62) TNFNOD2NOD1NOTUMLMNA
SCHEMBL7169094 0.75 TP53 (0.40) TNFNOD2NOD1LMNAMAPT
SCHEMBL6805438 0.74 ALDH1A1 (0.53) TNFNOD2NOD1NOTUMLMNA
SCHEMBL8567503 0.74 NOTUM (0.59) TNFNOD2NOD1NOTUMMAPT
SCHEMBL32673424 0.74 NOTUM (0.62) TNFNOD2NOD1NOTUMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825225-B2 useful against a number of human and veterinary pathogens, including gram-positive aerobic bacteria such as multiply-resistant staphylococci and streptococci, anaerobic organisms such as bacteroides and clostridia species, and acid-fast organisms PHARMACIA & UPJOHN COMPANY 2004-11-30 US disclosed
US-20040116413-A1 Novel bicyclic isoxazolinones as antibacterial agents PHARMACIA & UPJOHN COMPANY 2004-06-17 US disclosed