SCHEMBL6813012

SCHEMBL6813012

c1ccc(CCc2cc(OCc3ccccc3)ccc2N2CCCC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.53
LTA4H P09960 2/20 0.48
NPC1 O15118 1/20 0.46
CASP3 P42574 1/20 0.46
RAB9A P51151 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
MAOB P27338 2/20 0.46
ALOX5 P09917 1/20 0.45
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
MAOA P21397 1/20 0.44
CYP2D6 P10635 2/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28071588 0.86 LTA4H (0.48) HRH3LTA4HNPC1CASP3RAB9A
SCHEMBL25846133 0.80 HRH3 (0.49) HRH3LTA4HNPC1CASP3RAB9A
SCHEMBL17659705 0.79 HTR1A (0.54) HRH3LTA4HNPC1CASP3RAB9A
SCHEMBL17659018 0.78 HTR1A (0.52) HRH3LTA4HNPC1CASP3RAB9A
SCHEMBL8321069 0.77 RAB9A (0.50) HRH3LTA4HNPC1CASP3RAB9A
SCHEMBL11102792 0.76 HRH3 (0.53) HRH3NPC1RAB9AHTT
SCHEMBL8319330 0.76 NPC1 (0.52) HRH3LTA4HNPC1CASP3RAB9A
SCHEMBL6702208 0.74 LMNA (0.56) LTA4HMAOBALOX5HTR1ADRD2
SCHEMBL8322225 0.74 MAOB (0.58) HRH3LTA4HMAOBALOX5MAOA
SCHEMBL16046663 0.73 LTA4H (0.62) HRH3LTA4HNPC1CASP3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937458-B1 Pyrrolidine and piperidine derivatives HOFFMANN LA ROCHE (CH) 2004-12-29 EP disclosed