SCHEMBL6814243

SCHEMBL6814243

CNc1nc(NC)c2nc(-c3ccc(OC)cc3)c(-c3ccc(OC)cc3)nc2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.48
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 4/20 0.44
MAPT P10636 2/20 0.44
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
RXFP1 Q9HBX9 1/20 0.41
SYK P43405 2/20 0.41
DHFR P00374 1/20 0.40
NOS1 P29475 1/20 0.40
CHRNA7 P36544 1/20 0.40
MERTK Q12866 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SHMT2 P34897 1/20 0.39
ADORA2A P29274 2/20 0.38
ADORA2B P29275 1/20 0.38
TUBB4A P04350 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6811045 0.82 NOS1 (0.41) ADORA1ALDH1A1KDM4EMAPTLMNA
SCHEMBL6819013 0.82 NOS1 (0.56) ADORA1ALDH1A1KDM4EMAPTLMNA
SCHEMBL21852751 0.70 ALDH1A1 (0.67) ADORA1ALDH1A1KDM4EMAPTLMNA
SCHEMBL10456274 0.69 NOS1 (0.43) ADORA1KDM4ELMNATDP1NOS1
SCHEMBL6815719 0.69 CYP1A2 (0.43) ALDH1A1KDM4ELMNATDP1NOS1
SCHEMBL14525866 0.68 ALDH1A1 (0.64) ADORA1ALDH1A1KDM4EMAPTLMNA
SCHEMBL14983461 0.67 DHFR (0.56) ADORA1ALDH1A1KDM4EMAPTLMNA
SCHEMBL12067539 0.67 DHFR (0.56) ADORA1ALDH1A1KDM4EMAPTLMNA
SCHEMBL12131238 0.66 ALDH1A1 (0.53) ADORA1ALDH1A1KDM4EMAPTLMNA
SCHEMBL30696045 0.66 ALDH1A1 (0.53) ADORA1ALDH1A1KDM4EMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144412-B1 IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES 4 AZA BIOSCIENCE NV (BE) 2004-09-29 EP claimed