Picolamine

Picolamine

SCHEMBL6818607

Cc1c(=O)c(Cc2ccc(F)c(F)c2)cn2nc(C(=O)O)sc12.NCc1cccnc1

nearest known ligand 0.34

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.34
TBXAS1 P24557 5/20 0.33
S1PR3 Q99500 1/20 0.33
TRPA1 O75762 1/20 0.33
NR1D1 P20393 1/20 0.33
NR1H3 Q13133 1/20 0.33
VNN1 O95497 1/20 0.33
CXCR3 P49682 1/20 0.32
CACNA1G O43497 1/20 0.32
CACNA1H O95180 1/20 0.32
CACNA1I Q9P0X4 1/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2B Q13224 2/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
BLM P54132 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Niacinamide SCHEMBL6818598 0.89 FYN (0.39) PLA2G7VNN1CACNA1GCACNA1HCACNA1I
SCHEMBL6485426 0.89 P2RY14 (0.36) S1PR3CACNA1GCACNA1HCACNA1I
SCHEMBL6818605 0.86 ALDH1A1 (0.42) S1PR3TRPA1ALDH1A1LMNAMAPK1
SCHEMBL6477100 0.79 CHRM4 (0.43) S1PR3TRPA1CACNA1GCACNA1HCACNA1I
SCHEMBL6818812 0.73 CHRM4 (0.37) S1PR3TRPA1CACNA1GCACNA1HCACNA1I
SCHEMBL6813649 0.72 KDM5A (0.36) TBXAS1ALDH1A1
SCHEMBL6484565 0.69 RXRA (0.35) S1PR3TRPA1ALDH1A1LMNAMAPK1
SCHEMBL6476575 0.68 KDM5A (0.40) CACNA1HALDH1A1PTGDR2
SCHEMBL6813645 0.66 FYN (0.36) VNN1ALDH1A1
SCHEMBL6814009 0.66 PTGER4 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014908-A1 HETEROBICYLCIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed