SCHEMBL6819871

SCHEMBL6819871

CC1=C2CCc3ccccc3N2C(C)CC1=O

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 8/20 0.55
NOTUM Q6P988 3/20 0.41
ALDH1A1 P00352 1/20 0.39
OPRM1 P35372 2/20 0.37
OPRK1 P41145 2/20 0.37
OPRL1 P41146 2/20 0.37
ROCK1 Q13464 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6815716 0.77 ALDH1A1 (0.41) SRD5A1NOTUMALDH1A1ROCK1
SCHEMBL6822926 0.77 OPRM1 (0.43) SRD5A1NOTUMALDH1A1OPRM1OPRK1
SCHEMBL6820043 0.72 SRD5A1 (0.67) SRD5A1NOTUMALDH1A1OPRM1OPRK1
SCHEMBL6822784 0.71 SRD5A1 (1.00) SRD5A1
SCHEMBL11995386 0.66 ROCK1 (0.50) NOTUMALDH1A1ROCK1
SCHEMBL14733729 0.66 ROCK1 (0.50) NOTUMALDH1A1ROCK1
SCHEMBL15965528 0.66 ROCK1 (0.50) NOTUMALDH1A1ROCK1
SCHEMBL22005465 0.64 ROCK1 (0.51) NOTUMALDH1A1ROCK1
SCHEMBL7167355 0.64 SLC6A2 (0.44) NOTUMALDH1A1OPRM1OPRK1OPRL1
SCHEMBL7075121 0.64 ROCK1 (0.51) NOTUMALDH1A1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102765-B1 PROCESS FOR THE SYNTHESIS OF (1$i(H))-BENZO C]QUINOLIZIN-3-ONES DERIVATIVES APPLIED RESEARCH SYSTEMS (AN) 2003-09-17 EP claimed
US-6723850-B1 N-ALKYLATION OF THE THIOAMIDE WITH A VINYL KETONE IN PRESENCE OF A STRONG BASE; 6-CHLORO-(1H)-3,4-DIHYDROQUINOLIN-2-THIONE REACTED WITH ETHYL VINYL KETONE APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2004-04-20 US disclosed
EP-1102765-B1 PROCESS FOR THE SYNTHESIS OF (1$i(H))-BENZO C]QUINOLIZIN-3-ONES DERIVATIVES APPLIED RESEARCH SYSTEMS (AN) 2003-09-17 EP disclosed