SCHEMBL6823478

SCHEMBL6823478

Brc1ccc2c(c1)cc(-c1ccccc1)n2Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.52
NPC1 O15118 1/20 0.49
KRAS P01116 1/20 0.46
GRIK1 P39086 1/20 0.46
GRIK2 Q13002 1/20 0.46
CFTR P13569 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
PTGS2 P35354 2/20 0.43
ALDH1A1 P00352 2/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PDE6D O43924 1/20 0.41
ALDH2 P05091 1/20 0.41
ALDH3A1 P30838 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8762904 0.85 CCR2 (0.55) KRAS
SCHEMBL6820278 0.83 PTGS2 (0.53) GRIK1GRIK2PTGS2
SCHEMBL28387470 0.82 ESR1 (0.53) ESR1CFTRL3MBTL1PTGS2ALDH1A1
SCHEMBL4887683 0.82 L3MBTL1 (0.61) ESR1L3MBTL1PTGS2ALDH1A1PDE6D
SCHEMBL6822028 0.82 PTGS2 (0.58) GRIK1GRIK2L3MBTL1PTGS2ALDH1A1
SCHEMBL8761771 0.80 MAPK8 (0.59) PTGS2
SCHEMBL6823869 0.80 NPC1 (0.50) ESR1NPC1ALDH1A1
SCHEMBL8763754 0.79 POLB (0.46) NPC1KRASL3MBTL1ALDH1A1
SCHEMBL6821149 0.78 GRIK1 (0.75) GRIK1GRIK2ALDH1A1
SCHEMBL4415758 0.78 BRD4 (0.48) ESR1NPC1CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048331-A1 N-ARYLALKYL-3-AMINOALKOXYINDOLES AND THEIR USE AS 5-HT LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2004-06-10 WO disclosed