SCHEMBL6823942

SCHEMBL6823942

CC(=O)NCc1ccc(CN(NC(=O)O)C(=O)N2CCOCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
TPSAB1 Q15661 2/20 0.43
KMT2A Q03164 2/20 0.42
HTR2A P28223 3/20 0.41
HTR2C P28335 3/20 0.41
HTR2B P41595 3/20 0.41
USP2 O75604 2/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ESR1 P03372 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6823784 0.87 NOS3 (0.46) NOS3NOS1TPSAB1KMT2AHTR2A
SCHEMBL6823459 0.85 NPSR1 (0.44) TPSAB1KMT2AHTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL6820134 0.81 NOS3 (0.50) NOS3NOS1TPSAB1KMT2AHTR2A
SCHEMBL6823012 0.72 NPSR1 (0.42) TPSAB1KMT2AHTTALDH1A1
Hydrochloric Acid SCHEMBL7991650 0.71 ALDH1A1 (0.64) NOS3NOS1KMT2AUSP2HTT
SCHEMBL12133623 0.67 KMT2A (0.76) KMT2AALDH1A1KDM4E
SCHEMBL8602590 0.66 HRH3 (0.58) TPSAB1KMT2AALDH1A1
SCHEMBL19112444 0.66 KMT2A (0.54) KMT2AUSP2HTTKDM4E
Hydrochloric Acid SCHEMBL6823011 0.66 NPSR1 (0.43) TPSAB1KMT2AHTR2AHTR2CHTR2B
SCHEMBL7977518 0.66 KMT2A (0.59) TPSAB1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004067522-A1 AZAPHENYLALANINE DERIVATIVES AND THEIR USE AS ANTITHROMBOTIC AGENTS LEK PHARMACEUTICALS D.D. (SI) 2004-08-12 WO disclosed