SCHEMBL6824322

SCHEMBL6824322

Cc1ccc(C(=O)c2cccc(-c3cc(NCCCN(C)C)nc(N)n3)c2O)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.36
WNT1 P04628 1/20 0.35
DYRK1A Q13627 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
PIK3CD O00329 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HTT P42858 2/20 0.34
BRCA1 P38398 1/20 0.34
HIF1A Q16665 1/20 0.34
SYK P43405 1/20 0.34
CALCA P06881 1/20 0.34
HRH4 Q9H3N8 2/20 0.33
NUDT1 P36639 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TMEM97 Q5BJF2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6824329 0.85 HTT (0.36) TLR8PIM2PIK3CDSMN1; SMN2HTT
SCHEMBL6824771 0.74 CDK1 (0.38) TLR8HRH4ALDH1A1HPGDHSD17B10
SCHEMBL6821420 0.70 CDK1 (0.43) TLR8DYRK1AHRH4RAD52MEN1
SCHEMBL6923124 0.69 CDK1 (0.53) SMN1; SMN2HTTALDH1A1KMT2A
SCHEMBL12124182 0.67 HTT (0.62) SMN1; SMN2HTTALDH1A1HPGDTMEM97
SCHEMBL6824848 0.67 CACNA1G (0.43) HSD17B10KDM4E
SCHEMBL6820704 0.67 CDK1 (0.59) SMN1; SMN2HTTADORA2AADORA1ALDH1A1
SCHEMBL15757860 0.66 NUDT1 (0.54) TLR8PIK3CDHRH4NUDT1ADORA2A
SCHEMBL6823612 0.65 CDK1 (0.38) SMN1; SMN2HTTADORA2AADORA1HPGD
SCHEMBL15757276 0.65 NUDT1 (0.60) TLR8HRH4NUDT1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO claimed
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed