SCHEMBL6825032

SCHEMBL6825032

N#Cc1ccc([N+](=O)[O-])c(O)c1.N#Cc1cccc(O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 2/20 0.49
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
RECQL P46063 1/20 0.47
BLM P54132 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
GPR35 Q9HC97 1/20 0.46
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
EGFR P00533 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1142893 0.89 VCAM1 (0.59) VCAM1MAPTALDH1A1KDM4ELMNA
SCHEMBL31432469 0.89 VCAM1 (0.59) VCAM1MAPTALDH1A1KDM4ELMNA
SCHEMBL29566889 0.77
SCHEMBL51546 0.77
SCHEMBL1330201 0.77
SCHEMBL31326843 0.76 VCAM1 (0.64) VCAM1MAPTALDH1A1KDM4ELMNA
SCHEMBL103929 0.76 VCAM1 (0.64) VCAM1MAPTALDH1A1KDM4ELMNA
SCHEMBL7397116 0.75 ENPP2 (0.52) MAPTALDH1A1LMNACYP3A4HSD17B10
Hydrochloric Acid SCHEMBL28758837 0.75 ENPP2 (0.52) MAPTALDH1A1LMNACYP3A4HSD17B10
SCHEMBL7153973 0.74 GPR35 (0.58) VCAM1MAPTALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1185261-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-02-25 EP disclosed
EP-1185261-A1 IL-8 RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-03-13 EP disclosed
US-6262113-B1 HYDROXY- OR MERCAPTO-PHENYLUREAS SMITHKLINE BEECHAM CORPORATION 2001-07-17 US disclosed
WO-2000076495-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-21 WO disclosed