SCHEMBL6826385

SCHEMBL6826385

O=C(O)NC1CCC(=NOCc2ccccn2)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.43
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 1/20 0.42
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
ALOX5 P09917 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
CNR2 P34972 2/20 0.38
CNR1 P21554 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DRD4 P21917 1/20 0.38
GAA P10253 2/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6825996 0.83 CHRM2 (0.42) SIGMAR1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL6820957 0.82 ALDH1A1 (0.46) NPC1RAB9AALDH1A1CNR2CNR1
SCHEMBL6826045 0.81 SSTR4 (0.39) KDM4EALDH1A1CNR2CNR1GAA
SCHEMBL6820484 0.78 SYK (0.39) SIGMAR1SMN1; SMN2KDM4EALDH1A1DRD4
SCHEMBL7065633 0.78 SIGMAR1 (0.45) SIGMAR1SMN1; SMN2LMNAKDM4EALDH1A1
SCHEMBL6820130 0.74 SYK (0.38) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL27714486 0.71 SIGMAR1 (0.70) SIGMAR1SMN1; SMN2KDM4EALDH1A1CHRM2
SCHEMBL10843601 0.71 SMN1; SMN2 (0.44) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL25119945 0.69 L3MBTL1 (0.44) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL6825967 0.69 SYK (0.37) RAB9ASMN1; SMN2KDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004099185-A1 2-CYANOPYRROLIDINE DERIVATIVES AND THEIR USE AS DPP-IV INHIBITORS FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2004-11-18 WO disclosed
WO-2004048352-A2 2-CYANOPYRROLIDINES AND THEIR ANALOGUES AS DPP-IV INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-06-10 WO disclosed