SCHEMBL7065633

SCHEMBL7065633

O=C(O)NC1CCC(=NOCc2cccnc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.45
HDAC8 Q9BY41 1/20 0.43
HSD11B1 P28845 1/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP17A1 P05093 1/20 0.40
CYP19A1 P11511 1/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
NAPRT Q6XQN6 1/20 0.40
C3AR1 Q16581 1/20 0.39
FKBP1A P62942 2/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6820957 0.86 ALDH1A1 (0.46) ALDH1A1TSHR
SCHEMBL6826045 0.78 SSTR4 (0.39) KDM4EALDH1A1
SCHEMBL20357412 0.78 CHRM2 (0.50) SIGMAR1HSD11B1CYP17A1CYP19A1ALDH1A1
SCHEMBL6826385 0.78 SIGMAR1 (0.43) SIGMAR1KDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL6828166 0.77 HSD11B1 (0.40) HSD11B1KDM4ECYP17A1CYP19A1ALDH1A1
SCHEMBL20357434 0.76 CHRM2 (0.54) SIGMAR1HDAC8HSD11B1CYP17A1CYP19A1
SCHEMBL6825996 0.75 CHRM2 (0.42) SIGMAR1ALDH1A1LMNATSHRHTT
SCHEMBL6817016 0.74 CHRNB2 (0.41) HSD11B1KDM4ECYP17A1CYP19A1ALDH1A1
Hydrochloric Acid SCHEMBL6919466 0.73 DPP4 (0.51)
SCHEMBL6820894 0.72 KMT2A (0.52) HSD11B1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048352-A2 2-CYANOPYRROLIDINES AND THEIR ANALOGUES AS DPP-IV INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-06-10 WO disclosed