SCHEMBL6828649

SCHEMBL6828649

CC(C)c1cc(=O)[nH]nc1-c1sc(NC(=O)CCN2CCOCC2)nc1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
NPC1 O15118 1/20 0.48
TSHR P16473 1/20 0.48
CLK1 P49759 1/20 0.48
RAB9A P51151 1/20 0.48
TRPV4 Q9HBA0 2/20 0.44
CASR P41180 4/20 0.44
LMNA P02545 2/20 0.43
CYP2C19 P33261 1/20 0.43
TERT O14746 2/20 0.43
PTGS2 P35354 1/20 0.43
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
ADORA2A P29274 3/20 0.41
ADORA1 P30542 3/20 0.41
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6828984 0.85 ALK (0.47) ALDH1A1NPC1TSHRRAB9ATRPV4
Hydrochloric Acid SCHEMBL6828816 0.85 ALDH1A1 (0.47) ALDH1A1NPC1TSHRCLK1RAB9A
SCHEMBL6830910 0.84 ALDH1A1 (0.46) ALDH1A1TSHRLMNAMAPTKMT2A
Hydrochloric Acid SCHEMBL6828860 0.84 ALDH1A1 (0.47) ALDH1A1NPC1TSHRCLK1RAB9A
Hydrochloric Acid SCHEMBL6829009 0.83 HPGD (0.43) ALDH1A1NPC1TRPV4LMNAPTGS2
SCHEMBL6825783 0.82 ADORA1 (0.56) ALDH1A1TSHRMEN1MAPTKMT2A
SCHEMBL6828830 0.80 ADORA2A (0.48) ALDH1A1NPC1TSHRRAB9AMEN1
SCHEMBL6825903 0.79 HPGD (0.47) ALDH1A1TRPV4LMNACYP2C19PTGS2
SCHEMBL6830218 0.79 ALDH1A1 (0.43) ALDH1A1TSHRLMNAMEN1MAPT
SCHEMBL6830646 0.79 ADORA2A (0.53) ALDH1A1NPC1RAB9ALMNAGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed