SCHEMBL6828894

SCHEMBL6828894

CC(C)c1cc(=O)[nH]nc1-c1sc(NC(=O)c2cccc3ccccc23)nc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CNR1 P21554 1/20 0.44
XIAP P98170 2/20 0.43
ADORA3 P0DMS8 8/20 0.42
CNR2 P34972 1/20 0.42
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ADORA2A P29274 4/20 0.40
KDM4E B2RXH2 1/20 0.40
ADORA1 P30542 3/20 0.40
BCL2L1 Q07817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6828483 0.89 XIAP (0.44) SMN1; SMN2NPSR1XIAPADORA3ALDH1A1
SCHEMBL6828997 0.87 ADORA3 (0.49) SMN1; SMN2NPSR1XIAPADORA3ALDH1A1
SCHEMBL6826020 0.85 NPC1 (0.48) SMN1; SMN2NPSR1XIAPADORA3ALDH1A1
SCHEMBL6828357 0.84 ADORA2A (0.51) NPSR1XIAPADORA3NPC1RAB9A
SCHEMBL6830337 0.84 ADORA2A (0.50) SMN1; SMN2XIAPADORA3ALDH1A1NPC1
SCHEMBL6830646 0.81 ADORA2A (0.53) XIAPALDH1A1NPC1RAB9AADORA2A
SCHEMBL6825783 0.81 ADORA1 (0.56) XIAPADORA3ALDH1A1ADORA2AADORA1
SCHEMBL6828729 0.81 ADORA1 (0.57) SMN1; SMN2ADORA3ALDH1A1NPC1RAB9A
SCHEMBL6830676 0.81 ADORA2A (0.43) SMN1; SMN2NPSR1XIAPADORA3ALDH1A1
SCHEMBL6828670 0.80 XIAP (0.44) SMN1; SMN2NPSR1XIAPADORA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed