SCHEMBL6830337

SCHEMBL6830337

CC(C)c1cc(=O)[nH]nc1-c1sc(NC(=O)c2ccncc2)nc1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.50
ADORA1 P30542 9/20 0.50
ADORA3 P0DMS8 11/20 0.46
ADORA2B P29275 2/20 0.46
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
XIAP P98170 1/20 0.44
CHRM5 P08912 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
PARP1 P09874 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826020 0.89 NPC1 (0.48) ADORA2AADORA1ADORA3ALDH1A1NPC1
SCHEMBL6828729 0.88 ADORA1 (0.57) ADORA2AADORA1ADORA3ALDH1A1NPC1
SCHEMBL6828357 0.88 ADORA2A (0.51) ADORA2AADORA1ADORA3ADORA2BNPC1
SCHEMBL6830676 0.86 ADORA2A (0.43) ADORA2AADORA1ADORA3ALDH1A1NPC1
SCHEMBL6828483 0.85 XIAP (0.44) ADORA2AADORA1ADORA3ALDH1A1NPC1
SCHEMBL6828894 0.84 SMN1; SMN2 (0.44) ADORA2AADORA1ADORA3ALDH1A1NPC1
SCHEMBL6828972 0.83 TRPV4 (0.47) ADORA2AADORA1ADORA3KMT2ASMN1; SMN2
SCHEMBL6825783 0.83 ADORA1 (0.56) ADORA2AADORA1ADORA3ALDH1A1KMT2A
SCHEMBL6830646 0.83 ADORA2A (0.53) ADORA2AADORA1ALDH1A1NPC1RAB9A
SCHEMBL6828997 0.83 ADORA3 (0.49) ADORA2AADORA1ADORA3ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed