SCHEMBL6829307

SCHEMBL6829307

CC(C)c1cc(=O)[nH]nc1-c1sc(NC(=O)CCNCc2ccccn2)nc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.41
ADORA1 P30542 9/20 0.41
ALDH1A1 P00352 4/20 0.39
NPC1 O15118 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
XIAP P98170 3/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2B P29275 1/20 0.38
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DGAT1 O75907 1/20 0.36
NAMPT P43490 1/20 0.36
RORC P51449 1/20 0.36
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6830218 0.85 ALDH1A1 (0.43) ADORA2AADORA1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL6830910 0.83 ALDH1A1 (0.46) ADORA2AADORA1ALDH1A1KMT2AMAPT
SCHEMBL6828357 0.82 ADORA2A (0.51) ADORA2AADORA1NPC1KMT2AMAPT
SCHEMBL6825783 0.81 ADORA1 (0.56) ADORA2AADORA1ALDH1A1KMT2AMEN1
SCHEMBL6828830 0.81 ADORA2A (0.48) ADORA2AADORA1ALDH1A1NPC1KMT2A
Hydrochloric Acid SCHEMBL6828629 0.78 ALDH1A1 (0.41) ADORA2AADORA1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL6133691 0.77 ADORA2A (0.46) ADORA2AADORA1ALDH1A1NPC1KMT2A
SCHEMBL6828649 0.77 ALDH1A1 (0.49) ADORA2AADORA1ALDH1A1NPC1KMT2A
SCHEMBL6830337 0.77 ADORA2A (0.50) ADORA2AADORA1ALDH1A1NPC1KMT2A
Hydrochloric Acid SCHEMBL6828860 0.77 ALDH1A1 (0.47) ADORA2AADORA1ALDH1A1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed