SCHEMBL6832689

SCHEMBL6832689

CSc1ccc2cc(C(=O)N[C@H]3CCCC[C@H]3C(=O)NCC3(C#N)CC3)[nH]c2c1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.38
GHSR Q92847 9/20 0.35
F10 P00742 2/20 0.35
PYGL P06737 1/20 0.35
P2RX7 Q99572 1/20 0.34
KCNH2 Q12809 2/20 0.34
OPRM1 P35372 1/20 0.34
DRD4 P21917 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6838954 0.88 F10 (0.37) GHSRF10PYGLKCNH2OPRM1
SCHEMBL5260638 0.88 CTSK (0.50) CTSK
SCHEMBL6829592 0.87 NPC1 (0.48) KCNH2NPC1RAB9AKMT2A
SCHEMBL5255587 0.85 F10 (0.35) CTSKGHSRF10PYGLKCNH2
SCHEMBL6832876 0.85 GHSR (0.37) GHSRPYGL
SCHEMBL6833095 0.83 PYGL (0.42) GHSRPYGLOPRM1
SCHEMBL7070887 0.82 PYGL (0.42) GHSRPYGL
SCHEMBL5256902 0.81 F10 (0.43) F10DRD4NPC1RAB9AKMT2A
SCHEMBL5255596 0.80 DRD4 (0.36) CTSKF10DRD4
SCHEMBL6838957 0.80 DRD4 (0.36) CTSKF10DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6747053-B2 Heteroaryl nitriles ROCHE PALO ALTO LLC 2004-06-08 US disclosed