SCHEMBL6832876

SCHEMBL6832876

CS(=O)(=O)Nc1ccc2cc(C(=O)N[C@H]3CCCC[C@H]3C(=O)NCC3(C#N)CC3)[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 12/20 0.37
CYP2C9 P11712 1/20 0.36
NAMPT P43490 1/20 0.36
MMP2 P08253 1/20 0.35
MMP13 P45452 1/20 0.35
PYGL P06737 1/20 0.35
PLA2G7 Q13093 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6838954 0.86 F10 (0.37) GHSRPYGL
SCHEMBL6832689 0.85 CTSK (0.38) GHSRPYGL
SCHEMBL6829592 0.85 NPC1 (0.48)
SCHEMBL6833075 0.82 F10 (0.32) GHSRPYGL
SCHEMBL6833095 0.81 PYGL (0.42) GHSRPYGL
SCHEMBL5258079 0.81 PLA2G7 (0.35) CYP2C9NAMPTMMP2MMP13PLA2G7
SCHEMBL6839074 0.81 GHSR (0.41) GHSRPYGL
SCHEMBL5258087 0.81 PLA2G7 (0.35) CYP2C9NAMPTMMP2MMP13PLA2G7
SCHEMBL7070887 0.80 PYGL (0.42) GHSRPYGL
SCHEMBL14565630 0.78 MMP2 (0.38) CYP2C9NAMPTMMP2MMP13PLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6747053-B2 Heteroaryl nitriles ROCHE PALO ALTO LLC 2004-06-08 US disclosed