SCHEMBL6845264

SCHEMBL6845264

CONc1cc(NC(=O)c2ccc(C(C)C)cc2)ccn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.51
NPC1 O15118 2/20 0.51
BRAF P15056 1/20 0.48
DEGS1 O15121 1/20 0.48
TRPV1 Q8NER1 1/20 0.47
ROCK2 O75116 2/20 0.47
ROCK1 Q13464 2/20 0.47
TYK2 P29597 5/20 0.46
JAK2 O60674 2/20 0.46
JAK1 P23458 1/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
SIRT3 Q9NTG7 1/20 0.44
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL988281 0.90 ROCK2 (0.61) RAB9ANPC1BRAFROCK2ROCK1
SCHEMBL6845277 0.89 ROCK2 (0.44) RAB9ANPC1BRAFROCK2ROCK1
SCHEMBL987306 0.76 ROCK2 (0.65) RAB9ANPC1BRAFDEGS1ROCK2
SCHEMBL30192651 0.75 ROCK2 (0.77) RAB9ANPC1TRPV1ROCK2ROCK1
SCHEMBL6559116 0.75 ROCK2 (0.64) RAB9ANPC1BRAFROCK2ROCK1
SCHEMBL6845275 0.75 ROCK2 (0.47) RAB9ANPC1BRAFDEGS1TRPV1
SCHEMBL23844169 0.73 LMNA (0.76) RAB9ANPC1TRPV1ROCK2ROCK1
SCHEMBL19860113 0.72 NPC1 (0.76) RAB9ANPC1DEGS1TRPV1LMNA
SCHEMBL4609178 0.71 RAB9A (0.67) RAB9ANPC1KDM4ELMNATP53
SCHEMBL4609954 0.71 RAB9A (0.67) RAB9ANPC1KDM4ELMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7867999-B1 Hydroxyamino- and amino-substituted pyridine analogs for treating rho kinase-mediated diseases and conditions ALCON RESEARCH, LTD. (US) 2011-01-11 US disclosed