SCHEMBL6854322

SCHEMBL6854322

OCC#Cc1ccc(-c2ncccn2)s1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.41
MAPK14 Q16539 1/20 0.36
DPP4 P27487 1/20 0.35
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
GLA P06280 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
SLC5A2 P31639 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MELK Q14680 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869609 0.84 KDM4E (0.55) HDAC1ALDH1A1KDM4ENPC1GLA
SCHEMBL3904118 0.83 HDAC1 (0.38) HDAC1KDM4ENPC1GLAMAPT
SCHEMBL13722910 0.80 HDAC1 (0.36) HDAC1DPP4KDM4ENPC1GLA
SCHEMBL3900804 0.77 HDAC1 (0.41) HDAC1KDM4ENPC1GLAMAPT
SCHEMBL6847889 0.77 MAPK14 (0.51) HDAC1MAPK14DPP4KDM4EMAPT
SCHEMBL6879818 0.76 CYP2A6 (0.56) HDAC1MAPK14ALDH1A1
SCHEMBL6853750 0.76 MAPK14 (0.39) MAPK14DPP4ALDH1A1KDM4ENPC1
SCHEMBL6847879 0.76 MELK (0.37) MAPK14DPP4ALDH1A1KDM4ENPC1
SCHEMBL8013270 0.73 DPP4 (0.51) HDAC1MAPK14DPP4ALDH1A1KDM4E
SCHEMBL6880927 0.73 HDAC1 (0.41) HDAC1KDM4ENPC1GLAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed