SCHEMBL6857232

SCHEMBL6857232

O=c1[nH]c(C(F)(F)F)nc2c1N=C[N]2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.46
HCAR2 Q8TDS4 2/20 0.43
KDM5A P29375 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
HPGD P15428 5/20 0.36
ALDH1A1 P00352 4/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36
KDM4E B2RXH2 4/20 0.36
KHK P50053 1/20 0.36
RAD51 Q06609 1/20 0.35
MAPT P10636 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TSHR P16473 2/20 0.33
MEN1 O00255 2/20 0.33
POLB P06746 2/20 0.33
KMT2A Q03164 2/20 0.33
PABPC1 P11940 1/20 0.33
LMNA P02545 1/20 0.33
CRHBP P24387 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL142922 0.73 QTRT1 (0.42) MAPT
SCHEMBL546663 0.70 TYMS (0.40) ALDH1A1KDM4E
SCHEMBL546930 0.69 KDM4E (0.36) HPGDALDH1A1KDM4ELMNA
SCHEMBL5769223 0.65 PDE9A (0.38)
SCHEMBL10590403 0.64 NLRP3 (0.40) ALDH1A1HTTNPSR1KDM4EMAPT
SCHEMBL30388114 0.63 PKM (1.00) PKMHCAR2KDM5AKDM4CHPGD
SCHEMBL3118169 0.63 PKM (1.00) PKMHCAR2KDM5AKDM4CHPGD
SCHEMBL355917 0.61 ALDH1A1 (0.40) HPGDALDH1A1HTTKDM4ESMN1; SMN2
SCHEMBL2159691 0.60 PKM (0.59) PKMHCAR2KDM5AKDM4CHPGD
SCHEMBL7326945 0.60 TNKS (0.56) PKMHPGDALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383767-A1 TRIFLUOROMETHYLPURINES AS PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceutical Corporation (US) 2004-01-28 EP disclosed
WO-2002098878-A1 TRIFLUOROMETHYLPURINES AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2002-12-12 WO disclosed