SCHEMBL6861739

SCHEMBL6861739

COC(=O)CCCOc1ccc(C[C@H](NS(=O)(=O)c2ccc3ccccc3c2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
F2 P00734 5/20 0.48
PPARG P37231 2/20 0.46
PPARD Q03181 2/20 0.46
PPARA Q07869 2/20 0.46
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
KCNA5 P22460 1/20 0.43
CYSLTR1 Q9Y271 1/20 0.43
BACE1 P56817 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3441383 0.85 F2 (0.55) ALDH1A1F2BACE1MMP2MMP9
SCHEMBL6866437 0.82 ITGB3 (0.55) ALDH1A1ITGB3ITGA2BKCNA5MMP2
SCHEMBL6868246 0.81 ITGB3 (0.43) F2ITGB3ITGA2B
SCHEMBL6873358 0.81 TDP1 (0.46) ALDH1A1ITGB3ITGA2BKCNA5BACE1
SCHEMBL6862305 0.78 MMP2 (0.47) ALDH1A1PPARAITGB3ITGA2BKCNA5
SCHEMBL6861761 0.78 P2RX7 (0.45) F2ITGB3ITGA2BMMP2MMP9
SCHEMBL6870315 0.77 L3MBTL1 (0.52) ALDH1A1PPARGITGB3ITGA2BMMP2
SCHEMBL7984105 0.76 BACE1 (0.62) F2BACE1
SCHEMBL7983820 0.75 F2 (0.53) F2BACE1MMP2MMP9
SCHEMBL7983901 0.75 F2 (0.55) F2BACE1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1155003-B1 NOVEL GUANIDINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA GMBH (DE) 2004-08-11 EP disclosed
US-6340679-B1 FOR INHIBITING BONE RESORPTION, OSTEOPOROSIS, TUMOR GROWTH OR TUMOR METASTASIS, INFLAMMATION, OR FOR THE TREATMENT OF CARDIOVASCULAR DISORDERS, RESTENOSIS, ARTERIOSCLEROSIS, NEPHROPATHIES, RETINOPATHIES OR RHEUMATOID ARTHRITIS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-01-22 US disclosed
EP-1155003-A1 NOVEL GUANIDINE DERIVATIVES AS INHIBITORS OF CELL ADHESION Aventis Pharma Deutschland GmbH (DE) 2001-11-21 EP disclosed
WO-2000047564-A1 NOVEL GUANIDINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-17 WO disclosed
EP-1028114-A1 Novel guanidine derivatives as inhibitors of cell adhesion Aventis Pharma Deutschland GmbH (DE) 2000-08-16 EP disclosed