SCHEMBL6866437

SCHEMBL6866437

CC(C)(C)OC(=O)[C@H](Cc1ccc(OCCCC(=O)O)cc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.55
ITGA2B P08514 10/20 0.55
BCL2 P10415 1/20 0.52
MMP2 P08253 2/20 0.47
MMP9 P14780 2/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
MMP3 P08254 1/20 0.46
MMP13 P45452 1/20 0.46
KCNA5 P22460 2/20 0.45
CTSL P07711 1/20 0.45
CTSS P25774 1/20 0.45
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6862305 0.91 MMP2 (0.47) ITGB3ITGA2BBCL2MMP2MMP9
SCHEMBL6870315 0.90 L3MBTL1 (0.52) ITGB3ITGA2BBCL2MMP2MMP9
SCHEMBL6861761 0.87 P2RX7 (0.45) ITGB3ITGA2BBCL2MMP2MMP9
SCHEMBL7352181 0.83 ITGB3 (0.61) ITGB3ITGA2B
SCHEMBL6873358 0.83 TDP1 (0.46) ITGB3ITGA2BBCL2ALDH1A1MMP3
SCHEMBL6861739 0.82 ALDH1A1 (0.51) ITGB3ITGA2BMMP2MMP9ALDH1A1
SCHEMBL7488523 0.82 CA12 (0.56) ITGB3ITGA2BBCL2MMP2MMP9
SCHEMBL6868159 0.81 ITGB3 (0.51) ITGB3ITGA2BBCL2
SCHEMBL7342244 0.80 ITGB3 (0.62) ITGB3ITGA2B
SCHEMBL7489822 0.80 ITGB3 (0.61) ITGB3ITGA2BBCL2MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1155003-B1 NOVEL GUANIDINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA GMBH (DE) 2004-08-11 EP disclosed
US-6340679-B1 FOR INHIBITING BONE RESORPTION, OSTEOPOROSIS, TUMOR GROWTH OR TUMOR METASTASIS, INFLAMMATION, OR FOR THE TREATMENT OF CARDIOVASCULAR DISORDERS, RESTENOSIS, ARTERIOSCLEROSIS, NEPHROPATHIES, RETINOPATHIES OR RHEUMATOID ARTHRITIS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-01-22 US disclosed
EP-1155003-A1 NOVEL GUANIDINE DERIVATIVES AS INHIBITORS OF CELL ADHESION Aventis Pharma Deutschland GmbH (DE) 2001-11-21 EP disclosed
WO-2000047564-A1 NOVEL GUANIDINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-17 WO disclosed
EP-1028114-A1 Novel guanidine derivatives as inhibitors of cell adhesion Aventis Pharma Deutschland GmbH (DE) 2000-08-16 EP disclosed