SCHEMBL6863068

SCHEMBL6863068

Nc1cc(C(=O)NCC2CCCCC2)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.61
PDGFRB P09619 1/20 0.45
KDR P35968 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
F12 P00748 1/20 0.44
POLB P06746 1/20 0.44
HDAC6 Q9UBN7 1/20 0.42
CNR1 P21554 2/20 0.41
NPC1 O15118 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RAB9A P51151 1/20 0.41
HIF1A Q16665 1/20 0.41
CNR2 P34972 1/20 0.40
ADORA1 P30542 1/20 0.40
PANK1 Q8TE04 1/20 0.40
PANK3 Q9H999 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871382 0.91 ADORA2A (0.59) ADORA2AMEN1KMT2AF12NPC1
SCHEMBL6863385 0.86 MEN1 (0.47) ADORA2APDGFRBKDRMEN1KMT2A
SCHEMBL6868478 0.85 ADORA2A (0.64) ADORA2AKDRF12NPC1SMN1; SMN2
SCHEMBL6867628 0.81 ADORA2A (0.60) ADORA2AF12
SCHEMBL6870493 0.81 ADORA2A (0.40) ADORA2APDGFRBKDRMEN1KMT2A
SCHEMBL6870133 0.81 ADORA2A (0.59) ADORA2AKMT2AF12POLB
SCHEMBL6869989 0.80 ADORA2A (0.58) ADORA2AKDRF12NPC1SMN1; SMN2
SCHEMBL6869803 0.79 ADORA2A (0.41) ADORA2APDGFRBKDRMEN1KMT2A
SCHEMBL6869707 0.79 KIT (0.44) ADORA2APDGFRBKDRMEN1KMT2A
SCHEMBL6871448 0.79 ADORA2A (0.65) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed