SCHEMBL6869707

SCHEMBL6869707

Cc1ccc(-c2nc3cc(C(=O)NCC4CCCCC4)cc(N)n3n2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.44
ADORA2A P29274 5/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
METTL3 Q86U44 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
CHRM4 P08173 1/20 0.41
MMP13 P45452 1/20 0.41
KLKB1 P03952 1/20 0.40
MAOB P27338 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CA2 P00918 1/20 0.40
POLB P06746 1/20 0.39
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863790 0.91 KIT (0.46) KITADORA2ANPC1RAB9AMETTL3
SCHEMBL6870443 0.85 LMNA (0.45) KITADORA2AKDM4ENPC1ALDH1A1
SCHEMBL6871448 0.83 ADORA2A (0.65) KITADORA2ATDP1MMP13
SCHEMBL6863385 0.82 MEN1 (0.47) ADORA2ANPC1SMN1; SMN2MEN1KMT2A
SCHEMBL6871700 0.81 SMN1; SMN2 (0.41) ADORA2AKDM4ENPC1ALDH1A1HPGD
SCHEMBL6863351 0.80 PLAU (0.47) ADORA2AKDM4EALDH1A1HPGDCHRM4
SCHEMBL6863092 0.79 ADORA2A (0.64) ADORA2AMEN1KMT2A
SCHEMBL6869803 0.79 ADORA2A (0.41) ADORA2ATDP1MEN1KMT2ACA2
SCHEMBL6863068 0.79 ADORA2A (0.61) ADORA2ANPC1RAB9ASMN1; SMN2MEN1
SCHEMBL6870493 0.79 ADORA2A (0.40) KITADORA2AKDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed