SCHEMBL6868478

SCHEMBL6868478

Nc1cc(C(=O)NC2CCCCC2)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.64
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 3/20 0.49
LMNA P02545 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HTT P42858 1/20 0.45
GRM5 P41594 4/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TSHR P16473 1/20 0.41
KDR P35968 1/20 0.41
F12 P00748 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871382 0.86 ADORA2A (0.59) ADORA2ANPC1RAB9AF12HPGD
SCHEMBL6868095 0.85 KDM4E (0.53) ADORA2AKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL6863068 0.85 ADORA2A (0.61) ADORA2ASMN1; SMN2NPC1RAB9AKDR
SCHEMBL6863074 0.80 ADORA2A (0.62) ADORA2AKDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL6868483 0.80 ADORA2A (0.64) ADORA2AKDRF12
SCHEMBL6863748 0.80 ADORA2A (0.64) ADORA2AKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL6871945 0.80 ADORA2A (0.42) ADORA2AKDM4EALDH1A1LMNANPC1
SCHEMBL6867942 0.79 ADORA2A (0.71) ADORA2AKDM4EF12
SCHEMBL6869099 0.79 ADORA2A (0.98) ADORA2AF12HPGD
SCHEMBL6871467 0.79 ADORA2A (0.98) ADORA2AF12HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed