SCHEMBL6863385

SCHEMBL6863385

Nc1cc(C(=O)NCC2CCCCC2)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
POLB P06746 1/20 0.44
CNR1 P21554 1/20 0.44
NPC1 O15118 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDR P35968 2/20 0.43
PDGFRB P09619 1/20 0.43
AKT1 P31749 1/20 0.43
AKT2 P31751 1/20 0.43
PLK4 O00444 1/20 0.43
PDPK1 O15530 1/20 0.43
DAPK3 O43293 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
CHEK2 O96017 1/20 0.43
CDK1 P06493 1/20 0.43
RET P07949 1/20 0.43
PIM1 P11309 1/20 0.43
FGFR1 P11362 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863068 0.86 ADORA2A (0.61) MEN1KMT2APOLBCNR1NPC1
SCHEMBL6869803 0.86 ADORA2A (0.41) MEN1KMT2APOLBKDRPDGFRB
SCHEMBL6868095 0.84 KDM4E (0.53) MEN1KMT2ACNR1NPC1SMN1; SMN2
SCHEMBL6871448 0.82 ADORA2A (0.65) ADORA2A
SCHEMBL6869707 0.82 KIT (0.44) MEN1KMT2APOLBCNR1NPC1
SCHEMBL6863092 0.82 ADORA2A (0.64) MEN1KMT2AADORA2A
SCHEMBL6873157 0.81 HPGDS (0.51) KDRAKT1MAP4K4CHEK2CDK1
SCHEMBL6870493 0.81 ADORA2A (0.40) MEN1KMT2APOLBNPC1SMN1; SMN2
SCHEMBL6866973 0.78 BACE1 (0.48) KMT2APOLBNPC1SMN1; SMN2CAMK2D
SCHEMBL6871382 0.77 ADORA2A (0.59) MEN1KMT2ANPC1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed